Β1肾上腺素受体激动药

β1肾上腺素受体刺激劑(Beta1-adrenergic agonists)又名為 β1肾上腺素受体激动剂,是一種能選擇性作用於β1肾上腺素受体激动剂,β1肾上腺素受体刺激劑主要作用於心臟,通常由正腎上腺素激活。正腎上腺素則主要由交感神經的腎上腺素和循環全身的腎上腺素釋放而得。β1肾上腺素受体刺激劑激活後的效果主要為刺激心臟,例如:加速心率心肌收縮能力心導速率[1]

地诺帕明[2][3]多保他命扎莫特羅都屬於β1肾上腺素受体刺激劑。

文獻

  1. Sakuma, Tsutomu; Hida, Mieko; Nambu, Yoshihiro; Osanai, Kazuhiro; Toga, Hirohisa; Takahashi, Keiji; Ohya, Nobuo; Inoue, Masao; Watanabe, Yoh. . The Japanese Journal of Pharmacology (Japanese Pharmacological Society). 2001, 85 (2): 161–166. ISSN 0021-5198. doi:10.1254/jjp.85.161.
  2. Sakuma T, Hida M, Nambu Y, 等. . Jpn. J. Pharmacol. February 2001, 85 (2): 161–6. PMID 11286398. doi:10.1254/jjp.85.161.
  3. Nishio R, Matsumori A, Shioi T, 等. . J. Am. Coll. Cardiol. September 1998, 32 (3): 808–15. PMID 9741531. doi:10.1016/S0735-1097(98)00314-3.
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